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Falsodex (Fulvestrant)Complete info about Falsodex (Fulvestrant)Falsodex is an estrogen receptor antagonist, which has no agonist effects at all. It regulates down estrogen receptors (similiar to how Clen down regulates beta receptors, so you get decreased effects from the stuff). Basically, it binds to the Estrogen Receptor more strongly than tamoxifen, but still has no estrogen agonist effects. Here's the interesting part: the resultant down regulation of your estrogen receptors from the use of Falsodex results in decreased expression of the progesterone receptor as well! Tamoxifen, as we all know, can increase the sides from progesteronic drugs because of an increase in progesterone receptor expression. So you can take this stuff as both an anti-estrogen and an antiprogestin! No more buying Arimidex or whatever, and Bromocriptine! The stuff is administered via an IM injection of 250mgs once per month! And at that dose, it has most if not all of the same estrogen lowering effects of 1mg/day of Arim or 2.5mgs per day of Letrozole, but has the added benefits of lowering progesterone receptor expression. Falsodex is very hard to obtain anywhere on the black market, cost remain high, and availability low. References
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